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Drug Metabolism & Disposition

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Latest Articles

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    In Vitro Metabolism of 2-Methoxy-N-[3-[4-[3-methyl-4-[(6-methyl- 3-pyridinyl)oxy]anilino]-6-quinazolinyl]prop-2-enyl]acetamide (CP-724,714) by Aldehyde Oxidase and Predicting Its Percent Contribution Relative to CYP-Mediated Metabolism
    Kazuko Inoue, Kiyomi Kikuchi, Kazumi Takahashi, Seiji Hitaoka, Kazutomi Kusano and Takafumi Komori
    Drug Metabolism and Disposition August 2023, 51 (8) 962-969; DOI: https://doi.org/10.1124/dmd.122.000995
  • Open Access
    How Cryo-EM Has Expanded Our Understanding of Membrane Transporters
    Stefanie A. Baril, Tomoka Gose and John D. Schuetz
    Drug Metabolism and Disposition August 2023, 51 (8) 904-922; DOI: https://doi.org/10.1124/dmd.122.001004
  • Mass Balance and Absorption, Distribution, Metabolism, and Excretion Properties of Balcinrenone following Oral Administration in Combination with Intravenous Microtracer in Healthy Subjects
    Open Access
    Mass Balance and Absorption, Distribution, Metabolism, and Excretion Properties of Balcinrenone following Oral Administration in Combination with Intravenous Microtracer in Healthy Subjects
    Bo Lindmark, Xue-Qing Li, Chandrali Bhattacharya, Greggory Housler, Maria Heijer, Ryan A. Bragg, Malin Gränfors, Marta Pelay-Gimeno, Wouter H.J. Vaes, Somasekhara Menakuru, Patricia Ely Pizzato, Hans Ericsson and Susanne Johansson
    Drug Metabolism and Disposition August 2023, 51 (8) 995-1004; DOI: https://doi.org/10.1124/dmd.122.001240
  • METTL7A (TMT1A) and METTL7B (TMT1B) Are Responsible for Alkyl <em>S</em>-Thiol Methyl Transferase Activity in Liver
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    METTL7A (TMT1A) and METTL7B (TMT1B) Are Responsible for Alkyl S-Thiol Methyl Transferase Activity in Liver
    Drake A. Russell, Marvin K. Chau, Yuanyuan Shi, Ian N. Levasseur, Benjamin J. Maldonato and Rheem A. Totah
    Drug Metabolism and Disposition August 2023, 51 (8) 1024-1034; DOI: https://doi.org/10.1124/dmd.123.001268
  • Soy Protein Containing Diet Attenuates Murine Drug Exposure and Activity via Hepatic and Intestinal Cytochrome P450 Induction
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    Soy Protein Containing Diet Attenuates Murine Drug Exposure and Activity via Hepatic and Intestinal Cytochrome P450 Induction
    Jill M. Wetter, Rita Ciurlionis, Caitlin J. Krause, Michael J. Liguori, Christian Goess, Suzanne Mathieu and J. Cory Kalvass
    Drug Metabolism and Disposition August 2023, 51 (8) 1005-1015; DOI: https://doi.org/10.1124/dmd.123.001249
  • Assumptions Underlying Hepatic Clearance Models: Recognizing the Influence of Saturable Protein Binding on Driving Force Concentration and Discrimination Between Models of Hepatic Clearance
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    Assumptions Underlying Hepatic Clearance Models: Recognizing the Influence of Saturable Protein Binding on Driving Force Concentration and Discrimination Between Models of Hepatic Clearance
    Julia A. Schulz Pauly, Jin Wang, Colin J. Phipps and John Cory Kalvass
    Drug Metabolism and Disposition August 2023, 51 (8) 1046-1052; DOI: https://doi.org/10.1124/dmd.123.001326
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    Representative Rodent Models for Renal Transporter Alterations in Human Nonalcoholic Steatohepatitis
    Kayla L. Frost, Joseph L. Jilek, Erica L. Toth, Michael J. Goedken, Stephen H. Wright and Nathan J. Cherrington
    Drug Metabolism and Disposition August 2023, 51 (8) 970-981; DOI: https://doi.org/10.1124/dmd.122.001133
  • Open Access
    Systemic Exposure, Metabolism, and Elimination of [14C]-Labeled Amino Lipid, Lipid 5, after a Single Administration of mRNA Encapsulating Lipid Nanoparticles to Sprague-Dawley Rats
    Douglas Burdette, Lei Ci, Barclay Shilliday, Richard Slauter, Andrew Auerbach, Matthew Kenney, Örn Almarsson, Eugene Cheung and Tracy Hendrick
    Drug Metabolism and Disposition July 2023, 51 (7) 804-812; DOI: https://doi.org/10.1124/dmd.122.001194
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    Variants of Flavin-Containing Monooxygenase 3 Found in Subjects in an Updated Database of Genome Resources
    Miaki Makiguchi, Makiko Shimizu, Yuka Yokota, Erika Shimamura, Eiji Hishinuma, Sakae Saito, Masahiro Hiratsuka and Hiroshi Yamazaki
    Drug Metabolism and Disposition July 2023, 51 (7) 884-891; DOI: https://doi.org/10.1124/dmd.123.001310
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    The Disconnect in Intrinsic Clearance Determined in Human Hepatocytes and Liver Microsomes Results from Divergent Cytochrome P450 Activities
    Tashinga E. Bapiro, Scott Martin, Stephen D. Wilkinson, Alexandra L. Orton, Niresh Hariparsad, Stephanie Harlfinger and Dermot F. McGinnity
    Drug Metabolism and Disposition July 2023, 51 (7) 892-901; DOI: https://doi.org/10.1124/dmd.123.001323

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