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"Sequential Metabolism of AMG 487, a Novel CXCR3 Antagonist, Results in Formation of Quinone Reactive Metabolites That Covalently Modify CYP3A4 Cys239 and Cause Time-Dependent Inhibition of the Enzyme." Drug Metabolism and Disposition
40.7
(2012):
1429-1440.
Web. 18 April. 2024.