Substance | Intravenous | Oral | ||
---|---|---|---|---|
Urine | Feces | Urine | Feces | |
Total radioactivity | 5.2 | 92.9 | 2.8 | 94.5 |
Bosentan | 0.9 | 3.7 | 0.1 | 30.2 |
Ro 48-5033 | 1.9 | 47.5 | 1.1 | 34.6 |
Ro 64-1056 | 1.0 | 17.7 | 0.5 | 13.2 |
Ro 47-8634 | 0.2 | 6.4 | 0.1 | 6.7 |
Minor metabolites | 0.5 | 8.0 | 0.3 | 5.1 |
Unknown | 0.6 | 9.6 | 0.7 | 4.7 |
Data are presented in percent of dose administered.