Radiolabel | % of total radioactivity in urine | % of dose recovered in urine2-a |
---|---|---|
2-hydroxynevirapine glucuronide2-b | 22.9 | 18.6 |
3-hydroxynevirapine glucuronide2-b | 31.6 | 25.7 |
12-hydroxynevirapine glucuronide | 29.0 | 23.7 |
8-hydroxynevirapine glucuronide | 1.6 | 1.3 |
3-hydroxynevirapine | 1.5 | 1.2 |
12-hydroxynevirapine | 0.7 | 0.6 |
8-hydroxynevirapine | 1.6 | ND |
4-carboxynevirapine | 2.9 | 2.4 |
NVP | 3.3 | 2.7 |
Total | 90.7 | 76.2 |