Substrate | PON1 Type Q | PON1 Type R |
---|---|---|
pmol substrate hydrolyzed/min/mg PON1 | ||
Mevastatin | 485.1 ± 19.5 | 461.8 ± 23.1 |
Lovastatin | 489.6 ± 29.4 | 473.4 ± 18.9 |
Simvastatin | 684.5 ± 34.5 | 568.3 ± 11.7 |
Spironolactone | 234.8 ± 12.9 | 262.9 ± 10.5 |
The substrate concentration used was 5 μg/ml or 12.8, 12.4, 12.0, and 12.0 μM for mevastatin, lovastatin, simvastatin, and spironolactone, respectively. Each value represents the mean value of triplicate assays ± S.D.