Inhibitor | IC50 (μM) | |||
---|---|---|---|---|
Human | rCYP | |||
Bufuralol (n = 3)2-a | AMMC (n = 3)2-a | Bufuralol (n = 2) | AMMC (n = 2) | |
Quinidine | 0.06 ± 0.02 | 0.02 ± 0.01 | 0.02 | 0.01 |
Perhexiline | 0.4 ± 0.2 | 0.5 ± 0.1 | 0.5 | 0.3 |
Fluoxetine | 1.2 ± 0.8 | 1.2 ± 0.1 | 2.3 | 0.8 |
Norfluoxetine | 1.0 ± 0.2 | 1.5 ± 0.3 | 5 | 1 |
Quinine | 15 ± 3 | 4 ± 1 | —2-b | —2-b |
Dextromethorphan | 30 ± 10 | 9 ± 2 | 8 | 2 |
Imipramine | 35 ± 5 | 11 ± 3 | 13 | 4 |
Sparteine | >100 | 80 ± 10 | >100 | 40 |