BALC (Ring Methyl Oxidation) | ET (N-Deethylation) | |||||
---|---|---|---|---|---|---|
Km | Vmax | CLint | Km | Vmax | CLint | |
μM | nmol/mg protein/min | 10−6/mg protein/min | μM | nmol/mg protein/min | 10−6/mg protein/min | |
HLM | 67.6 ± 4.2b | 12.9 ± 1.6a b | 191.5 ± 15.4b | 842.5 ± 49.9b | 20.5 ± 3.4a | 24.4 ± 5.1b |
RLM | 38.3 ± 0.2a | 17.6 ± 1.2a | 461.3 ± 23.5a | 214.3 ± 26.1a | 19.2 ± 2.8a | 89.5 ± 10.9a |
MLM | 43.4 ± 0.6a b | 6.8 ± 1.4b | 156.8 ± 23.8b | 660.6 ± 59.5b | 14.5 ± 2.9a | 21.7 ± 3.9b |
MLM1-150 | 42.6 ± 13.6a b | 16.4 ± 3.4a | 385.1 ± 52.6a | 630.9 ± 128.0b | 22.9 ± 2.9a | 38.3 ± 5.1b |
Means in the same column followed by the same letter are not significantly different (P < 0.01). Values are the mean ± S.E.M. (n = 3).
↵1-150 DEET treated animals LD10 (200 mg/kg/day).