Control | Troleandomycin | GG918 | Cyclosporine | |
---|---|---|---|---|
Tacrolimus | ||||
AUC (ng/ml · min)a | 2,260 ± 430 | 5,200 ± 2,470* | 1,730 ± 270* | 4,390 ± 2,080* |
AUCM (ng/ml · min)a | 22,900 ± 10,900 | 72,100 ± 7,900* | 12,100 ± 4,500 | 70,200 ± 27,200* |
AUCM/AUCb | 9.35 ± 1.94 | 10.3 ± 2.4 | 6.24 ± 1.74 | 11.9 ± 2.1 |
Felodipine | ||||
AUC (ng/ml · min) | 4,380 ± 320 | 6,150 ± 900* | 4,000 ± 50 | 5,310 ± 950 |
AUCMc | 693 ± 38 | 3,120 ± 890* | 1,190 ± 110* | 1,520 ± 670 |
AUCM/AUCc | 0.158 ± 0.007 | 0.504 ± 0.116* | 0.297 ± 0.024* | 0.285 ± 0.116* |