Transporter | Substrate | Reference |
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abst or ibat Ileal sodium-dependent bile acid transporter | Taurocholate | Schneider et al. 1995; Craddock et al., 1998 |
Pept1 Oligopeptide transporter 1 | Aminocephalosporins, β-amino lactam antibiotics (cyclacillin, cephalexin, cephradine), acetylcholinesterase inhibitors (benazepril, quinapril), bestatin, renin inhibitors | Fei et al., 1994 |
Mct1 Monocarboxylic acid transporter 1 | Lactate and pyruvate transport (simple aryl and alkyl acids) | |
Oatp3 Intestinal organic anion transporting polypeptide 3 | Taurocholate, estrone sulfate | Walters et al., 2000 |
NPT1 Sodium-dependent phosphate tranporter 1 | Fosfomycin, foscarnet | Tsuji and Tamai, 1989 |
OCT1 Organic cation transporter 1 | Spermine, spermidine | |
Folic acid transporter | Methotrexate | |
CNT Nucleoside transporters N1 (purine) and N2 (pyrimidine) | Zidovudine, stavudine, thymidine, ribavirin, allopurinol, 5-fluorouracil | |
Amino acid carrier | d- and l-Methionine, l-methyldopa, baclofen, taurine, alanine | |
MDR1 or Pgp Multidrug resistance protein 1 or P-glycoprotein | Daunomycin, rhodamine 123, verapamil, diltiazem, colchicine, digoxin, quinidine, vincristine, etoposide β-blockers (sotalol, pafenolol, celiprolol, tanilol) | |
Mrp2 Multidrug resistance-associated protein 2 | Glutathione conjugates, glucuronide conjugates, leukotriene C4, vincristine | Gotoh et al., 2000; Mottino et al., 2000 |
BCRP Breast cancer resistance protein | Topotecan, mitoxantrone, anthracyclines | Doyle et al., 1998; Zamber et al., 2003 |
Mrp3 |
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Rost et al., 2002
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