IC50 summary of UGT2B7 in the presence of different inhibitors
Inhibitor | IC50 | Hill Constant |
|---|---|---|
| mM | n | |
| Naloxone | 0.135 ± 0.033 | 0.53 ± 0.07 |
| Valproic acid | 0.711 ± 0.390 | 0.29 ± 0.06 |
| Codeine | 3.03 ± 0.76 | 0.94 ± 0.27 |
| Ibuprofen | 0.975 ± 0.193 | 1.90 ± 0.62 |
| Morphine | 0.591 ± 0.266 | 0.42 ± 0.08 |
| Diclofenac | 0.059 ± 0.010 | 0.93 ± 0.11 |