TABLE 3

Single dose pharmacokinetic parameters for total radioactivity in female rats (n = 4)


Parameter

Female Rat
Cmax (μg Eq/ml) 6.91 ± 0.54
Tmax (h) 24 ± 0.0
AUC0-∞ (h · μg Eq/ml) 1038.0 ± 64.4
t1/2 (h) 91.8 ± 5.6
Vd (ml) 259.1 ± 25.8
CLp (ml/h)
1.95 ± 0.11