Inactivator | Kinetic Parameters | Reference | ||
---|---|---|---|---|
kinact | KI | |||
min-1 | μM | |||
Amprenavir | 0.45 | 0.64 | ||
0.60 | 0.37 | Ernest et al. (2003) | ||
Diclofenac | N.D. | N.D. | ||
0.26 | 1600 | Masubuchi et al. (2002) | ||
Diltiazem | 0.012 | 0.48 | ||
0.015 | 1 | Dai et al. (2003) | ||
Erythromycin | 0.072 | 15.2 | ||
0.081 | 9.9 | Dai et al. (2003) | ||
Raloxifene | 0.36 | 18.7 | ||
0.16 | 9.9 | Chen et al. (2002) | ||
Troleandomycin | 0.032 | 2.4 |
|
N.D., not determined.