Inhibitor | Ki | ||||
---|---|---|---|---|---|
Supersomes | HLM | RECO | |||
μM | |||||
Benzbromarone | 0.004 | 0.011 | 0.11 | ||
Diclofenac | 1.6 | 2.9 | 9.3 | ||
Fluvoxamine | 0.63 | 5.7 | 6.6 | ||
Gemfibrozil | 12.4 | 0.98 | 13.9 | ||
(S)-Ibuprofen | 4.3 | 3.2 | 17.1 | ||
Indomethacin | 53.4 | 12.8 | 48.7 | ||
Ketoconazole | 0.38 | 2.1 | 2.4 | ||
Miconazole | 0.028 | 0.038 | 0.11 | ||
Phenytoin | 5.6 | 10.2 | 11.1 | ||
Piroxicam | 0.47 | 9.8 | 6.7 | ||
Sulfaphenazole | 0.06 | 0.15 | 1.3 | ||
Tolbutamide | 1.5 | 3.5 | 2.0 |