Drug | Pretreatment | Binding Parameter (±S.E.)a | ||||||||
---|---|---|---|---|---|---|---|---|---|---|
Bmax | Kd | BNS | Kp max | Kp min | ||||||
μM | μM | |||||||||
Imipramine | None | 11 ± 3.2 | 6.3 ± 4.6 | 0.77 ± 0.23 | 360 ± 120 | 150 ± 23 | ||||
ABT | 9.7 ± 3.6 | 6.2 ± 5.7 | 1.1 ± 0.31 | 380 ± 110 | 160 ± 29 | |||||
Propranolol | None | 66 ± 39 | 36 ± 18 | 0.41 ± 0.11 | 240 ± 46 | 69 ± 6.8 | ||||
| ABT | 89 ± 17 | 62 ± 9.9 | 0.30 ± 0.14 | 180 ± 19 | 63 ± 11 |
↵ a Using eq. 3.