Compound | kinact | KI | kinact/KI | References |
---|---|---|---|---|
min−1 | μM | min−1 mM−1 | ||
D-617 | 0.07 | 7.9 | 9 | Wang et al. (2004) |
N-Desmethyltamoxifen | 0.13 | 12.0 | 11 | |
Fluvoxamine | 0.05 | 3.7 | 13 | |
Fluoxetine | 0.04 | 2.3 | 17 | Mayhew et al. (2000) |
Nortriptyline | 0.04 | 2.1 | 19 | |
Nefazodone | 0.27 | 12.5 | 22 | |
Clarithromycin | 0.23 | 4.1 | 56 | Mayhew et al. (2000) |
Tamoxifen | 0.03 | 0.5 | 59 | Zhao et al. (2002) |
R-Verapamil | 0.39 | 6.5 | 60 | Wang et al. (2004) |
N-Desmethylerythromycin | 0.34 | 5.7 | 60 | |
Erythromycin | 0.17 | 2.3 | 75 | |
14-OH-clarithromycin | 0.05 | 0.5 | 102 | |
Amlodipine | 0.35 | 2.6 | 135 | |
Nicardipine | 0.18 | 1.2 | 149 | |
Norverapamil | 1.12 | 5.9 | 190 | Wang et al. (2004) |
N-Desmethyldiltiazem | 0.29 | 1.5 | 200 | Mayhew et al. (2000) |
S-Verapamil | 0.64 | 3.0 | 215 | Wang et al. (2004) |
Lopinavir | 0.1 | 0.4 | 244 | Ernest et al. (2005) |
Propoxyphene | 0.41 | 1.4 | 293 | |
Nelfinavir | 0.22 | 0.5 | 458 | Ernest et al. (2005) |
Diltiazem | 0.17 | 0.4 | 472 | Jones et al. (1999) |
SKF-525A | 0.25 | 0.4 | 625 | |
Triacetyloleandomycin | 0.11 | 0.1 | 1222 | |
Mifepristone | 0.67 | 0.4 | 1634 | |
Saquinavir | 0.31 | 0.2 | 1824 | Ernest et al. (2005) |
Amprenavir | 0.73 | 0.3 | 2808 | Ernest et al. (2005) |
Ritonavir | 0.32 | 0.1 | 3200 | Ernest et al. (2005) |