[11C]Verapamil | [11C]GR205171 | [18F]Altanserin | |||||||
---|---|---|---|---|---|---|---|---|---|
SUVincrease | Kp,increase | SUVincrease | Kp,increase | SUVincrease | Kp,increase | ||||
Cerebellum | |||||||||
Rat | 4.1* | 5.8** | 3.6** | 3.5** | 2.6*a | 2.3*a | |||
Rat low dose CsA | 1.4ns | 1.5** | |||||||
Guinea pig | 3.9*** | 2.9** | 2.3** | 2.0ns | |||||
Minipigb | 1.8 | 0.8 | |||||||
Monkeyb | 4.3 | 3.6 | 2.1 | 2.5 | |||||
High binding regionc | |||||||||
Rat | 2.6*a | 2.9*a | |||||||
Minipigb | 2.0 | 0.9 | |||||||
Monkeyb |
|
| 2.6 | 2.9 |
|
|