Compound and Conc. | Papp(A-B) | Papp(B-A) | Efflux Ratio |
---|---|---|---|
× 10−6 cm/s | |||
[14C]Sorafenib, 0.1 μM | 16.4 ± 12.3 | 76.6 ± 21.2 | 4.67 ± 3.73 |
[14C]Sorafenib, 1 μM | 33.5 ± 16.1 | 83.8 ± 8.60 | 2.50 ± 1.23 |
Ketoprofen, 2 μM | 26.4 ± 6.68 | 18.3 ± 3.98 | 0.694 ± 0.320 |
Metoprolol, 2 μM | 32.5 ± 2.44 | 24.6 ± 3.02 | 0.756 ± 1.09 |
Fluvastatin, 2 μM | 17.5 ± 1.95 | 23.6 ± 2.16 | 1.35 ± 0.194 |
Atenolol, 10 μM | 0.662 ± 0.0480 | 0.860 ± 0.250 | 1.30 ± 0.389 |
Digoxin, 10 μM | 0.370 ± 0.0552 | 22.0 ± 3.53 | 59.5 ± 13.0 |