TABLE 1
Potencies for active compounds from primary qHTS across assays
Curve classes 1.1, 1.2, 2.1, and 2.2.
Potency
hPXR
hPXR LBD
CYP3A4 Induction
rPXR
μ
M
<1
8
8
13
9
1–10
124
98
86
79
10–32
178
88
113
87