Donor | mRNA | |||||
---|---|---|---|---|---|---|
Rifampicin | Carbamazepine | Estradiol | ||||
EC50 (μM) | Emax (fold increase) | EC50mM (μM) | Emax (fold increase) | EC50 (μM) | Emax (fold increase) | |
mRNA | ||||||
Hu1399 | 0.45 | 7.7 | 9.4 | 11.5 | 1.7 | 12.7 |
Hu8127 | 1.4 | 24 | 18 | 15 | 2.5 | 33 |
Hu4069 | 1.1 | 19 | 51 | 28 | 1.6 | 57 |
Mean of all donors | 0.98 ± 0.49 | 16.9 ± 8.4 | 26 ± 22 | 18.2 ± 8.7 | 1.9 ± 0.5 | 34 ± 22 |
Activity | ||||||
Hu1399 | 0.66 | 4.7 | 74 | 5.6 | 1.6 | 2.2 |
Hu8127 | 2.0 | 30 | 160 | 33 | 8.8 | 44 |
Hu4069 | 1.3 | 16 | 202 | 26 | 1.9 | 16 |
Mean of all donors | 1.3 ± 0.7 | 16.9 ± 12.7 | 145 ± 65 | 21.5 ± 14.3 | 4.1 ± 4.1 | 20 ± 21 |