Metabolites | Human | ||
---|---|---|---|
Urinea | Feces | Total | |
Ertugliflozin | 1.5 ± 0.4 | 33.8 ± 6.8 | 35.3 ± 7.0 |
M1 | 0.7 ± 0.3 | 1.7 ± 0.8 | 2.4 ± 0.7 |
M2 | 0.4 ± 0.3 | 1.0 ± 0.5 | 1.4 ± 0.6 |
M3 | N.D. | 1.4 ± 0.3 | 1.4 ± 0.3 |
M4a | 5.7 ± 1.7 | N.D. | 5.7 ± 1.7 |
M4b | 1.9 ± 0.4 | N.D. | 1.9 ± 0.4 |
M4c | 31.7 ± 7.0 | N.D. | 31.7 ± 7.0 |
M5a | 1.2 ± 0.6 | N.D. | 1.2 ± 0.6 |
M5b | 3.4 ± 1.0 | N.D. | 3.4 ± 1.0 |
N.D., not detected.
↵a Urine pooled from 0 to 48 hours.