Compound | OATP1B1 | OATP1B3 | OATP2B1 | NTCP | ||||
---|---|---|---|---|---|---|---|---|
IC50 | Ki | IC50 | Ki | IC50 | Ki | IC50 | Ki | |
ยตM | ||||||||
Atazanavir | 0.96 | 0.42 | 17 | 7.3 | >40 | >30 | >40 | >40 |
Cyclosporine | 1.5 | 0.66 | 3.1 | 1.3 | >18 | >13 | 4.8 | 4.8 |
Gemfibrozil | 130 | 58 | >1000 | >420 | 770 | 570 | 89 | 89 |
Lopinavir | 0.77 | 0.34 | >10 | >4.2 | >10 | >7.4 | >10 | >10 |
Rifampicin | 5.0 | 2.2 | 190 | 82 | >630 | >470 | >630 | >630 |