Mean | CV | Range | Range of max/min | No. of samples | Q | Degrees of freedom | P value | I2 | Heterogeneity | References | |
---|---|---|---|---|---|---|---|---|---|---|---|
fmol/μg protein | % | fmol/μg protein | fmol/μg protein | % | |||||||
Human liver tissue | |||||||||||
OATP1B1 | 5.9 | 42.5 | 0.8–44.3 | 3.3–6.6 | 86 | 10.30 | 4 | <0.05 | 61 | Moderate | Balogh et al. (2012), Kimoto et al. (2012), Karlgren et al. (2012), Prasad et al. (2014), Vildhede et al. (2014) |
OATP1B3 | 2.0 | 45.2 | 0.1–11.8 | 1.5–32 | 86 | 20.60 | 4 | <0.001 | 81 | High | Balogh et al. (2012), Kimoto et al. (2012), Karlgren et al. (2012), Prasad et al. (2014), Vildhede et al. (2014) |
OATP2B1 | 1.9 | 39.8 | 0.6–5.4 | 1.5–7.5 | 86 | 26.64 | 4 | <0.001 | 85 | High | Balogh et al. (2012), Kimoto et al. (2012), Karlgren et al. (2012), Prasad et al. (2014), Vildhede et al. (2014) |
Sandwich-cultured human hepatocytes | |||||||||||
OATP1B1 | 5.8 | 51.5 | 2.4–11.3 | 4.7a | 5 | — | — | — | — | — | Kimoto et al. (2012), Bi et al. (2012) |
OATP1B3 | 0.8 | 30.0 | 0.5–1.2 | 2.5a | 5 | — | — | — | — | — | Kimoto et al. (2012), Bi et al. (2012) |
OATP2B1 | 1.0 | 16.0 | 0.8–1.2 | 1.5a | 5 | — | — | — | — | — | Kimoto et al. (2012), Bi et al. (2012) |
Human cryopreserved hepatocytes in suspension | |||||||||||
OATP1B1 | 4.2 | 24.1 | 0.2–7.0 | 3.0a | 17 | — | — | — | — | — | Kimoto et al. (2012), Prasad et al. (2014), Bi et al. (2012), Ji et al. (2012), Kunze et al. (2014) |
OATP1B3 | 1.8 | 26.8 | 0.005–5.8 | 3.6a | 17 | — | — | — | — | — | Kimoto et al. (2012), Prasad et al. (2014), Bi et al. (2012), Ji et al. (2012), Kunze et al. (2014) |
OATP2B1 | 1.6 | 28.3 | 0.022–4.1 | 3.6a | 17 | — | — | — | — | — | Kimoto et al. (2012), Prasad et al. (2014), Bi et al. (2012), Ji et al. (2012), Kunze et al. (2014) |
—–, Not applicable
↵a Based on data reported in Kimoto et al. (2012)