N-Desethyl sunitinib (1a) | Yes (expected) | Yes (expected) | Yes (expected) | Yes (expected) |
Trovafloxacin glucuronide (2a) | Yes (expected) | Yes (n.d.) | Yes (expected) | Yes (expected) |
4-Oxo-carbazeran (3a) | Yes (expected) | Yes (n.d.) | No (expected) | No (n.d.) |
2-Oxo-zoniporide (4a) | Yes (expected) | Yes (n.d.) | Yes (unexpected)a | Yes (expected) |
4-Hydroxytolbutamide (5a) | Yes (expected) | Yes (n.d.) | No (expected) | Yes (n.d.) |
N-Acetylprocainamide (6a) | Yes (expected) | Yes (n.d.) | Yes (unexpected)b | Yes (expected) |
Trifluoperazine-N-glucuronide (7a) | Yes (n.d.)c | Yes (n.d.) | No (n.d.) | No (expected) |