Enzyme Source | Hydrolase Activity | RAF | Contribution | ||||||||
---|---|---|---|---|---|---|---|---|---|---|---|
Indiplon | Fenofibrate | Procaine | Prasugrel | AADAC | CES1 | CES2 | AADAC | CES1 | CES2 | Total | |
pmol/min/mg protein | nmol/min/mg protein | nmol/min/mg protein | nmol/min/mg protein | % | % | % | % | % | % | % | |
AADAC | 265.0 | 136.7 | |||||||||
CES1 | 84.0 | 19.2 | |||||||||
CES2 | 4.3 | 40.2 | |||||||||
HIM | 221.0 | 0 | 11.1 | 225.1 | 0.83 | 0 | 2.60 | 50.6 | 0 | 46.4 | 97.0 |
HLM | 338.3 | 421.4 | 2.3 | 304.5 | 1.28 | 5.01 | 0.54 | 57.3 | 31.6 | 7.1 | 96.0 |