Assay Test Compound | Concentration Range | IC50 | Maximum % Inhibition |
---|---|---|---|
Assay 1 | µM | µM | |
Abiraterone acetate | 0.03–30.0 | 3.0 | 83 |
Abiraterone | 0.03–30.0 | 2.9 | 59 |
Quercetin | 0.03–30.0 | 1.3 | 96 |
Assay 2 | |||
Abiraterone sulfate | 0.005–5.0 | 0.044 | 97 |
Abiraterone sulfate N-oxide | 0.03–30.0 | 5.4 | 81 |
Quercetin | 0.03–30.0 | 3.3 | 95 |