Treatment | Km,app | Vmax |
---|---|---|
µM | nmol/min/mg protein | |
Tamoxifen to NDM | ||
Vehicle | 3.8 ± 0.9 | 0.78 ± 0.02 |
Rifampin | 4.3 ± 1.3 | 2.6 ± 0.8* |
Tamoxifen to 4OHT | ||
Vehicle | 7.9 ± 2.8 | 0.84 ± 0.17 |
Rifampin | 7.8 ± 1.5 | 0.85 ± 0.26 |
NDM to endoxifen | ||
Vehicle | 5.9 ± 1.1 | 2.0 ± 0.72 |
Rifampin | 6.7 ± 1.4 | 1.9 ± 0.64 |
4OHT to endoxifen | ||
Vehicle | 13 ± 3.3 | 0.35 ± 0.10 |
Rifampin | 9.9 ± 2.8 | 2.6 ± 0.53* |
↵* P < 0.05 relative to vehicle.