Transporter | Protein Expression | Percent Coefficient of Variation |
---|---|---|
Uptake | ||
OAT1 | 5.33 ± 1.88 | 35.3 |
OAT2 | 0.93 ± 0.32 | 34.6 |
OAT3 | 3.50 ± 1.55 | 44.3 |
OAT4 | 0.52 ± 0.23 | 44.5 |
OCT2 | 7.42 ± 2.84 | 38.3 |
OCTN1 | 1.27 ± 0.59 | 46.1 |
OCTN2 | 0.57 ± 0.24 | 41.2 |
SGLT2 | 3.67 ± 1.86 | 50.6 |
Efflux | ||
P-gp | 2.09 ± 0.82 | 39.3 |
BCRP | < LLOQ | |
MRP2 | 1.35 ± 0.63 | 46.4 |
MRP4 | 0.91 ± 0.64 | 70.7 |
MATE1 | 5.06 ± 2.27 | 45.0 |
MATE2-K | < LLOQ |