Substrate | Hepatocyte Format | Hepatocyte Lot | Km | Vmax | Vmax/Km | RAF |
---|---|---|---|---|---|---|
µM | pmol/min per milligram | µl/min per milligram | ||||
E3S | Suspension | HUP1001 | 1.14 | 77.63 | 67.9 | 0.68 |
HUP1001 (rifamycin SV) | 0.93 | 166.2 | 179.3 | 1.95 | ||
HUM122D | 0.53 | 114.8 | 218.2 | 2.43 | ||
HUM4122D (rifamycin SV) | 0.32 ± 0.032 | 84.4 ± 6.5 | 269 ± 48 | 3.02 ± 0.55 | ||
SCHH | HU1651 | 0.7 | 84.8 | 121 | 1.16 | |
HUM4122D | 1.25 | 141.8 | 113.1 | 1.18 | ||
HUM4122D (rifamycin SV) | 0.52 | 56 | 108 | 1.12 | ||
CCK-8 | Suspension | HUP1001 | NCa | NC | 0.71b | 0.04 |
HUM122D | 1.2 | 6.8 | 5.8 | 0.31 | ||
SCHH | HU1651 | 1.9 | 3.0 | 1.6 | 0.09 | |
HUM4122D | 1.3 | 7.6 | 5.9 | 0.31 | ||
TCA | Suspension | HUP1001 | 23.6 | 437 | 18.5 | 0.23 |
HUM122D | 21.4 | 246 | 11.5 | 0.14 | ||
SCHH | HU1651 | 12.9 | 594.3 | 45.9 | 0.57 | |
HUM4122D | 25.6 | 577.1 | 22.6 | 0.28 |