Condition | TC50 (μM) | Reference | |
---|---|---|---|
PrestoBlue assay | ciPTEC–OAT1 2D (24 h) | 212 ± 11 | |
ciPTEC–OAT1 2D (48 h) | 85 ± 9 | ||
RS (24 h) | 97 ± 8 | ||
RS (48 h) | 93 ± 5 | ||
Live/Dead assay | RS (24 h) | 11.0 ± 3.0 | |
RS (48 h) | 5.5 ± 2.0 | ||
Literature | ciPTEC–OAT1 2D (24 h) | 114 ± 25 | Nieskens et al., 2016 |
ciPTEC–OAT1 2D (48 h) | 189 ± 48 | ||
ciPTEC–OAT1 2D (72 h) | 223 ± 67 | ||
CHO-hOAT1 (24 h) | 21 ± 7 | Cihlar et al. (2009) | |
HEK-293–OAT1 (24 h) | 10 ± 2 | Zhang et al. (2015) |
HEK–OAT1, human embryonic kidney cells 293 overexpressing OAT-1.