Drug | IC50 | IC50 Fold Shift | |
---|---|---|---|
Without 30-Minute Preincubation | With 30-Minute Preincubation | ||
µM | µM | ||
Cyclosporine A | 21.6 ± 4.5 | 0.43 ± 0.12 | 50.2 |
Quinidine | 7.7 ± 0.9 | 4.5 ± 0.7 | 1.7 |
Pyrimethamine | 1.8 ± 0.2 | 1.3 ± 0.1 | 1.4 |
Ritonavir | 2.2 ± 0.3 | 1.1 ± 0.1 | 2.0 |
Trimethoprim | 9.6 ± 1.2 | 9.2 ± 0.7 | 1.1 |