TABLE 1
Time dependence of the inhibitory effect of azamulin on CYP3A4/5
Preincubation Time (min)
IC
50
± S.E. (µM)
0
1.0 ± 0.1
10
0.46 ± 0.02
100
0.20 ± 0.02
220
0.13 ± 0.01