TABLE 4

Summary of transporters involved in transporting selected compounds in human

The uptake and efflux transporters of each selected compounds are summarized from Drug Interaction Solution Database, University of Washington (https://didb.druginteractionsolutions.org).

CompoundOATPsOATsOther transporters
Rosuvastatin1A2, 1B1, 1B3, 2B1OAT3NTCP, BCRP, MRP1-5, P-gp
Cerivastatin1B1, 1B3, 2B1P-gp, BCRP, MRPs
Fluvastatin1B1, 1B3, 2B1NTCP, BCRP, MRP2, P-gp
Pitavastatin1A2, 1B1, 1B3, 2B1NTCP, BCRP, MRP3, MRP4, P-gp
Atorvastatin1A2, 1B1, 1B3, 2B1NTCP, BCRP, MRP1, MRP2, MRP4, P-gp
Sorafenib1B1, 1B3OCT1, MRP2, P-gp
Pravastatin1A2, 1B1, 1B3, 2B1OAT3, OAT4, OAT7NTCP, BCRP, MRP1, MRP2, MRP4, MRP5, BSEP, P-gp
Danoprevir1B1, 1B3MRP2, P-gp
Maraviroc1B1P-gp
Bosentan1B1, 1B3, 2B1MRP2, P-gp
Repaglinide1B1, 1B3P-gp
Grazoprevir1B1, 1B3BCRP, P-gp
Telmisartan1B3, 2B1
Asunaprevir1B1, 2B1P-gp
Valsartan1B1, 1B3OAT1, OAT3MRP2, P-gp