TABLE 2

Percentage of revefenacin and its metabolites identified in pooled plasma after a single intravenous dose of 20 μg [14C]-revefenacin (n = 6) and an oral dose of 200 μg [14C]-revefenacin (n = 6)

[14C]-revefenacin, [14C]-labeled revefenacin.

Circulating Radioactivity (%) IntravenousCirculating Radioactivity (%) Oral
Revefenacin52.113.1
THRX-195518 (M2)14.312.5
THRX-697795 (M10)4.7912.5
THRX-193305 (M9)2.812.93
THRX-609075 (M1)1.663.63
THRX-177860 (M8)1.583.69