TABLE 5

Enzyme degradation rate

CYP IsoformKdeg (min−1)Reference
CYP1A20.00030(Faber and Fuhr, 2004)
CYP2B60.00036(Renwick et al., 2000)
CYP2C80.00053(Backman et al., 2009)
CYP2C90.00011(Renwick et al., 2000)
CYP2C190.00044
CYP2D60.00023(Liston et al., 2002; Venkatakrishnan and Obach, 2005)