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Using the Dynamic Well-stirred Model to Extrapolate Hepatic Clearance of OATP Substrates without Assuming Albumin-Mediated Hepatic Drug Uptake
Zhengyin Yan, Li Ma, Nicky Hwang, Julie Huang, Jane R. Kenny and Cornelis E.C.A. Hop
Drug Metabolism and Disposition April 11, 2024, DMD-AR-2024-001645; DOI: https://doi.org/10.1124/dmd.124.001645