Synthesis and SAR of aminothiazole fused benzazepines as selective dopamine D2 partial agonists
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Acknowledgments
The authors would like to thank Jennifer Van Anda, James Hall, John McCauley, Xiaomei Ye, Timothy Blake, Don Pivonka and Russ Spreen for analytical chemistry support; Leonard Tini, Cindy Shen, William Potts, James Bulgarelli, Patricia Schroeder and Bernard Lanoue for DMPK support; JianWei Liu, Linda Sygowski and John Zysk for neuroscience binding and functional assay support and My Linh Do and Zeke Zeller for behavioral pharmacology support. We wish to thank Håkan Wikström for excellent
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