Evidence for the interaction of imatinib at the transport-substrate site(s) of the multidrug-resistance-linked ABC drug transporters ABCB1 (P-glycoprotein) and ABCG2

Leukemia. 2008 Feb;22(2):445-7. doi: 10.1038/sj.leu.2404897. Epub 2007 Aug 9.
No abstract available

Publication types

  • Letter
  • Research Support, N.I.H., Intramural
  • Comment

MeSH terms

  • ATP Binding Cassette Transporter, Subfamily B
  • ATP Binding Cassette Transporter, Subfamily B, Member 1 / metabolism*
  • ATP Binding Cassette Transporter, Subfamily G, Member 2
  • ATP-Binding Cassette Transporters / metabolism*
  • Adenosine Triphosphate / metabolism
  • Benzamides
  • Binding Sites
  • Drug Resistance, Multiple
  • Humans
  • Imatinib Mesylate
  • Neoplasm Proteins / metabolism*
  • Piperazines / metabolism*
  • Pyrimidines / metabolism*

Substances

  • ABCB1 protein, human
  • ABCG2 protein, human
  • ATP Binding Cassette Transporter, Subfamily B
  • ATP Binding Cassette Transporter, Subfamily B, Member 1
  • ATP Binding Cassette Transporter, Subfamily G, Member 2
  • ATP-Binding Cassette Transporters
  • Benzamides
  • Neoplasm Proteins
  • Piperazines
  • Pyrimidines
  • Imatinib Mesylate
  • Adenosine Triphosphate