Metabolism of tamoxifen by rat liver microsomes: formation of the N-oxide, a new metabolite

Biochem Pharmacol. 1980 Jul 1;29(13):1977-9. doi: 10.1016/0006-2952(80)90116-1.
No abstract available

MeSH terms

  • Animals
  • Biotransformation
  • Dealkylation
  • Hydrogen-Ion Concentration
  • Hydroxylation
  • In Vitro Techniques
  • Male
  • Microsomes, Liver / metabolism*
  • Oxidation-Reduction
  • Oxides / metabolism
  • Rats
  • Tamoxifen / metabolism*

Substances

  • Oxides
  • Tamoxifen