2024
- December: Special Section on Challenges and Opportunities in Application of Physiologically Base Pharmacokinetics Models
- November: Special Section on New and Emerging Areas and Technologies in Drug Metabolism and Disposition, Part II
- August: Special Section on Mechanisms of Drug Metabolism in Acetaminophen-Induced Hepatotoxicity
- June: Special Section on Cytochrome P450 Enzymes in Toxicology and as Drug Targets
2023
- October: New and Emerging Areas and Technologies in Drug Metabolism and Disposition, Part I
- September: Mechanism-Based Predictive Methods in Drug Discovery and Development
- August: Perspective on Drug Metabolism and Disposition, Part II
- June: Perspective on Drug Metabolism and Disposition, Part I
- March: Drug Metabolism and Precision Medicine
- February: Xenobiotic Receptors
- January: 50th Anniversary Celebration Collection
2022
- October: Mechanistic and Translational Research on Transporters in Toxicology
- September: New Era of Transporter Science: Unraveling the Functional Role of Orphan Transporters
- July: Drug Metabolism and Regulation
- June: Pharmacokinetics and ADME of Biological Therapeutics
- May: Drug Metabolism in Liver Injury and Repair
- April: Bile Acids, Drug Metabolism, and Toxicity
- January: ADME Databases
2020
- October: Natural Products
2019